Intermediates
Commercial
| Indication | Product Name | CAS No. | Structure |
|
Losartan |
2-Butyl-4-chloro-5-formylimidazole;BCFI | 83857-96-9 |  |
| Telmisartan | 2-n-propyl-4-methyl-6-(1-methylbenzimidazole-2-ylbenzimidazole);BIM | 152628-02-9 |  |
| Rivaroxaban | 4-(4-aminophenyl)morpholin-3-one | 438056-69-0 |  |
| 5-Chlorothiophene-2-carbonyl chloride | 42518-98-9 |  |
|
| 5-Chlorothiophene-2-carboxylic Acid | 24065-33-6 |  |
|
| (S)-N-Glycidylphthalimide | 161596-47-0 |  |
|
| 2-[[(5S)-2-Oxo-3-[4-(3-oxo-4-morpholinyl)phenyl]-5-oxazolidinyl]methyl]-1H-isoindole-1,3(2H)-dione | 446292-08-6 |  |
|
| (S)-4-(4-(5-(AMinoMethyl)-2-oxooxazolidin-3-yl)phenyl)Morpholin-3-one hydrochloride | 898543-06-1 |  |
|
Dabigatran Etexilate Mesilate |
N-(4-Cyano-Phenyl)-Glycine | 42288-26-6 |  |
| 4-Methylamino-3-nitro benzoic acid | 41263-74-5 |  |
|
| N-Ethyl 3-(pyridin-2-ylamino)propanoate | 103041-38-9 |  |
|
| 3-(3-amino-4-(methylamino)-N-(pyridin-2-yl)benzamido)propanoate | 212322-56-0 |  |
|
| Benazepril | 3-Bromo-2,3,4,5-tetrahydro-2H-benzo[b]azepin-2-one | 86499-96-9 |  |
| Sildenafil | 4-amino-1-methyl-3-propyl-1H-pyrazole-5-carboxamide hydrochloride | 247584-10-7 |  |
| Arotinolol | 5-(2-sulfanylidene-3H-1,3-thiazol-4-yl)thiophene-2-carboxamide | 52560-89-1 |  |
| Dronedarone |
(2-Butyl-5-nitrobenzofuran-3-yl)(4-hydroxyphenyl)methanone | 141645-16-1 |  |
| (2-butyl-5-nitrobenzofuran-3-yl)(4-(3-(dibutylaMino)propoxy)phenyl)Methanone | 141645-23-0 |  |
|
| Baricitinib | 2-(1-(ethylsulfonyl)azetidin-3-ylidene)acetonitrile | 1187595-85-2 |  |
| 7-((2-(triMethylsilyl)ethoxy)Methyl)-4-chloro-7H-pyrrolo[2,3-d]pyriMidine | 941685-26-3 |  |
|
| 4-(1H-Pyrazol-4-yl)-7-((2-(trimethylsilyl)ethoxy)methyl-7H-pyrrolo[2,3-d]pyrimidine | 941685-27-4 |  |
|
| [4-(1H-Pyrazol-4-yl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl]methyl pivalate | 1146629-77-7 |  |
|
| Celecoxib | 4'-Methylacetophenone | 122-00-9 |  |
| 4-Hydrazinobenzene-1-sulfonamide hydrochloride | 17852-52-7 |  |
|
| 4,4,4-Trifluoro-1-(p-tolyl)-1,3-butanedione | 720-94-5 |  |
|
| Isavuconazole | 2-Bromo-4'-cyanoacetophenone | 20099-89-2 |  |
| Deucravacitinib | Methyl 4,6-dichloropyridazine-3-carboxylate | 372118-01-9 |  |
| 2-methoxy-3-(1-methyl-1H-1,2,4-triazol-3-yl)aniline | 1609394-10-6 |  |
|
| Salbutamol | alpha-[(benzyl-tert-butylamino)methyl]-m-xylene-4,alpha,alpha'-triol | 24085-03-8 |  |
| Olaparib | 3-Bromo-4-fluorobenzaldehyde | 77771-02-9 |  |
| 3-Cyano-4-fluorobenzaldehyde | 218301-22-5 |  |
|
| 2-Fluoro-5-[(3-oxo-1(3H)-isobenzofuranylidene)methyl]-benzonitrile | 763114-25-6 |  |
|
| Netupitant | 6-(4-Methylpiperazin-1-yl)-4-(2-methylphenyl)nicotinamide | 342417-01-0 |  |
| 2-(3,5-bis(trifluoroMethyl)phenyl)-2-Methyl propanoic acid | 289686-70-0 |  |
|
| N-Methyl-4-(2-methylphenyl)-6-(4-methyl-1-piperazinyl)-3-pyridinamine Oxalic acid | 290297-25-5 |  |
|
| Pazopanib |
N-(2-chloropyriMidin-4-yl)-N,2,3-triMethyl-2H-indazol-6-aMine | 444731-75-3 |  |
| 2,3-dimethyl-2H-indazol-6-amine hydrochloride | 635702-60-2 |  |
|
| Oxcarbazepine |
10-Methoxy Iminostilbene (10-MISB) | 4698-11-7 |  |
| Iminodibenzyl（IDB） | 494-19-9 |  |
|
| Carbamazepine |
Dibenz[b,f]azepine-5-carbonyl chloride（ISBCC） | 33948-22-0 |  |
| Iminostilbene（ISB） | 256-96-2 |  |
|
| Baclofen | 3-(4-Chlorophenyl)glutaric acid | 35271-74-0 |  |
| Tapentadol Hydrochloride | 3’-Methoxypropiophenone;3-MPP | 37951-49-8 |  |
| Tramadol hydrochloride | 3-Bromoanisole;MBA | 2398-37-0 |  |
| Vonoprazan Fumarate |
5-(2-Fluorophenyl)-1H-pyrrole-3-carbaldehyde | 881674-56-2 |  |
| yridine-3-sulfonyl chloride | 16133-25-8 |  |
Under R&D
| Indication | Product Name | CAS No. | Structure |
|
Rimegepan |
(6S,9R)-6-(2,3-Difluorophenyl)-6,7,8,9-tetrahydro-9-[[tris(1-methylethyl)silyl]oxy]-5H-cyclohepta[b]pyridin-5-one | 1190363-46-2 |  |
| 2-Oxo-1-(4-piperidinyl)-2,3-dihydro-1H-imidazo[4,5-b]pyridine dihydrochloride | 781649-84-1 |  |
|
| 1-(1-(1H-imidazole-1-carbonyl)piperidin-4-yl)-1H-imidazo[4,5-b]pyridin-2(3H)-one | 1373116-06-3 |  |
|
| Upadacitinib | (3R,4S)-3-(2-Bromoacetyl)-4-ethyl-1-pyrrolidinecarboxylic acid phenylmethyl ester | 1428243-26-8 |  |
| Carbamic acid,N-[5-[(4-methylphenyl)sulfonyl]-5H-pyrrolo[2,3-b]pyrazin-2-yl]-, ethyl este | 1869118-24-0 |  |
|
Ubrogepant |
(3S,5S,6R)-3-amino-6-methyl-5-phenyl-1-(2,2,2-trifluoroethyl)piperidin-2-one hydrochloride | 1375470-88-4 |  |
| (3'S)-1',2',5,7-Tetrahydro-2'-oxospiro[6H-cyclopenta[b]pyridine-6,3'-[3H]pyrrolo[2,3-b]pyridine]-3-carboxylic acid | 1375541-21-1 |  |
